99% Tianeptine sodium paʻakai CAS 30123-17-2
Hōʻike
MEA | KANAWAI | HUA |
Ka nana aku | Pauda keʻokeʻo a melemele | ʻO ka pauka kristal keʻokeʻo |
Ka hikiwawe | Hiki ke hoʻoheheʻe ʻia i ka wai a methanol a me dichloromethane | Kūlike |
ʻIkepili | Na IR, E hoʻohālikelike me ka hana maʻamau | Kūlike |
(2) Hāʻawi ia i ka hopena o ka sodium | Kūlike | |
Na mea haumia A | ≤0.1% | ʻAʻole ʻike ʻia |
Pūhui pili | Kekahi Max hoʻokahi haumia≤0.1% | 0.060% |
Huina haumia≤0.4% | 0.36% | |
Nā mea hoʻoheheʻe koena (GC) | Acetidin≤ 0.5% | ND |
Dichloromethane≤ 0.06% | ND | |
Methanol≤ 0.3% | ND | |
Acetone≤ 0.5% | 0.29% | |
Acetonitrile≤0.041% | 0.022% | |
Ethanol≤0.5% | ND | |
N, N-dimethylformamide≤0.088% | ND | |
Wai | ≤ 5.0% | 3.8% |
ʻIke (HPLC) | 99.0%-101.0% (Ma ka anhydrousbasis) | 99.70% |
Palapala noi
ʻO ka sodium Tianeptinepaʻakaihe tricyclic antidepressant.He ʻokoʻa kona ʻano hana antidepressant mai ka tricyclic antidepressants kahiko.Hiki iā ia ke hoʻonui i ka reuptake o 5-HT i ka synaptic cleft.Nā hopena o ka HT neuronal conduction.ʻAʻohe pili no ka choline a i ʻole adrenergic receptors.ʻOi aku ka maikaʻi o ka antidepressant me ka tricyclics, akā ʻoi aku ka maikaʻi o ka hoʻomanawanui ma mua o ka tricyclics.No ka mālama ʻana i ke kaumaha haʻahaʻa, haʻahaʻa a koʻikoʻi paha, neurogenic a reactive depression, hopohopo a me ke kaumaha me ke kino, ʻoi aku ka ʻeha o ka ʻōpū, a me ka hopohopo a me ke kaumaha i nā mea maʻi e hilinaʻi ana i ka waiʻona i ka wā o ka haʻalele ʻana.